TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 8.10nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of human recombinant MAOB by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of human recombinant MAOB by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Inhibition of human recombinant MAOB by spectrophotometricallyMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibition of human recombinant MAOB by spectrophotometricallyMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 180nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 217nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 220nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 270nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 320nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 420nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 450nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR overexpressed in human SHEP cells after 75 mins by liquid scintillation spectrometric analy...More data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Inhibition of human recombinant MAOB by spectrophotometricallyMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 680nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 710nMAssay Description:Inhibition of MAOB in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 910nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in SH-EP1 cellsMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 970nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in SH-EP1 cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 980nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 1.49E+3nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 1.53E+3nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+3nMAssay Description:Inhibition of human recombinant MAOB by spectrophotometricallyMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 2.17E+3nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 2.17E+3nMAssay Description:Inhibition of MAOA in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 2.23E+3nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of human recombinant MAOB by spectrophotometricallyMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+3nMAssay Description:Inhibition of human recombinant MAOA by spectrophotometricallyMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 2.50E+3nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in SH-EP1 cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 2.56E+3nMAssay Description:Inhibition of MAOB in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 3.00E+3nMAssay Description:Displacement of [3H]cytisine from human alpha4beta2 nAChR expressed in SH-EP1 cellsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 3.40E+3nMAssay Description:Inhibition of MAOB in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 3.42E+3nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 3.69E+3nMAssay Description:Inhibition of MAOA in rat brain mitochondrial suspensionMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 3.78E+3nMAssay Description:Inhibition of MAOA in rat brain mitochondriaMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
University of Chile
Curated by ChEMBL
University of Chile
Curated by ChEMBL
Affinity DataKi: 3.80E+3nMAssay Description:Displacement of [125I]alpha-bungarotoxin from human alpha7 nAChR overexpressed in human SH-SY5Y cells after 120 mins by liquid scintillation spectrom...More data for this Ligand-Target Pair